A bridge for industrial and academic collaborations, this book overviews the concepts and therapeutic application of allosteric modulation to control protein function - explaining why it has gained strong momentum in drug discovery, technologies and methodologies to discover allosteric modulators, and allosteric modulator compounds.- Collects into one single resource the details on allosteric modulation of key drug targets, making for an encyclopedic coverage from basics to drug discovery applications- Describes methods to detect and analyze allosterism- Lets readers compare how allosteric modulators function and used across different platforms- Includes the major drug target classes with demonstrated allosteric modulation- Features a companion website with color images and protocols that readers can access